β-Tosylethylamine: A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams

Darren DiPietro; Robert M. Borzilleri; Steven M. Weinreb

doi:10.1021/jo00099a006

β-Tosylethylamine: A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams

Darren DiPietro
, Robert M. Borzilleri
, Steven M. Weinreb

Chemistry

Research output: Contribution to journal › Article › peer-review

32 Scopus citations

Abstract

Readily prepared β-tosylethylamine (3) can be used to synthesize N-tosylethyl (TSE)-protected amido compounds and β-lactams, which can be deprotected under mild conditions with potassium tert-butoxide.

Original language	English (US)
Pages (from-to)	5856-5857
Number of pages	2
Journal	Journal of Organic Chemistry
Volume	59
Issue number	20
DOIs	https://doi.org/10.1021/jo00099a006
State	Published - Oct 1 1994

All Science Journal Classification (ASJC) codes

Organic Chemistry

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10.1021/jo00099a006

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title = "β-Tosylethylamine: A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams",

abstract = "Readily prepared β-tosylethylamine (3) can be used to synthesize N-tosylethyl (TSE)-protected amido compounds and β-lactams, which can be deprotected under mild conditions with potassium tert-butoxide.",

author = "Darren DiPietro and Borzilleri, \{Robert M.\} and Weinreb, \{Steven M.\}",

year = "1994",

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journal = "Journal of Organic Chemistry",

issn = "0022-3263",

publisher = "American Chemical Society",

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T1 - β-Tosylethylamine

T2 - A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams

AU - DiPietro, Darren

AU - Borzilleri, Robert M.

AU - Weinreb, Steven M.

PY - 1994/10/1

Y1 - 1994/10/1

N2 - Readily prepared β-tosylethylamine (3) can be used to synthesize N-tosylethyl (TSE)-protected amido compounds and β-lactams, which can be deprotected under mild conditions with potassium tert-butoxide.

AB - Readily prepared β-tosylethylamine (3) can be used to synthesize N-tosylethyl (TSE)-protected amido compounds and β-lactams, which can be deprotected under mild conditions with potassium tert-butoxide.

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UR - https://www.scopus.com/pages/publications/0028034612#tab=citedBy

U2 - 10.1021/jo00099a006

DO - 10.1021/jo00099a006

M3 - Article

AN - SCOPUS:0028034612

SN - 0022-3263

VL - 59

SP - 5856

EP - 5857

JO - Journal of Organic Chemistry

JF - Journal of Organic Chemistry

IS - 20

ER -

β-Tosylethylamine: A Useful Reagent for Preparation of N-Protected Amides, Carbamates, and Related Compounds. Application to Synthesis of β-Lactams

Abstract

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