Mitsunobu reactions of n-alkyl and n-acyl sulfonamides-an efficient route to protected amines

James R. Henry; Lawrence R. Marcin; Matthias C. McIntosh; Paul M. Scola; G. Davis Harris; Steven M. Weinreb

doi:10.1016/S0040-4039(00)76177-6

Mitsunobu reactions of n-alkyl and n-acyl sulfonamides-an efficient route to protected amines

James R. Henry, Lawrence R. Marcin, Matthias C. McIntosh, Paul M. Scola, G. Davis Harris, Steven M. Weinreb

Chemistry

Research output: Contribution to journal › Article › peer-review

226 Scopus citations

Abstract

N-Methyl p-toluenesulfonamide and N-BOC p-toluenesulfonamide can be directly coupled with primary and secondary alcohols under Mitsunobu conditions to afford various sulfonamide-protected amines.

Original language	English (US)
Pages (from-to)	5709-5712
Number of pages	4
Journal	Tetrahedron Letters
Volume	30
Issue number	42
DOIs	https://doi.org/10.1016/S0040-4039(00)76177-6
State	Published - 1989

All Science Journal Classification (ASJC) codes

Biochemistry
Drug Discovery
Organic Chemistry

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10.1016/S0040-4039(00)76177-6

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title = "Mitsunobu reactions of n-alkyl and n-acyl sulfonamides-an efficient route to protected amines",

abstract = "N-Methyl p-toluenesulfonamide and N-BOC p-toluenesulfonamide can be directly coupled with primary and secondary alcohols under Mitsunobu conditions to afford various sulfonamide-protected amines.",

author = "Henry, {James R.} and Marcin, {Lawrence R.} and McIntosh, {Matthias C.} and Scola, {Paul M.} and {Davis Harris}, G. and Weinreb, {Steven M.}",

year = "1989",

doi = "10.1016/S0040-4039(00)76177-6",

language = "English (US)",

volume = "30",

pages = "5709--5712",

journal = "Tetrahedron Letters",

issn = "0040-4039",

publisher = "Elsevier Ltd",

number = "42",

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TY - JOUR

T1 - Mitsunobu reactions of n-alkyl and n-acyl sulfonamides-an efficient route to protected amines

AU - Henry, James R.

AU - Marcin, Lawrence R.

AU - McIntosh, Matthias C.

AU - Scola, Paul M.

AU - Davis Harris, G.

AU - Weinreb, Steven M.

PY - 1989

Y1 - 1989

N2 - N-Methyl p-toluenesulfonamide and N-BOC p-toluenesulfonamide can be directly coupled with primary and secondary alcohols under Mitsunobu conditions to afford various sulfonamide-protected amines.

AB - N-Methyl p-toluenesulfonamide and N-BOC p-toluenesulfonamide can be directly coupled with primary and secondary alcohols under Mitsunobu conditions to afford various sulfonamide-protected amines.

UR - http://www.scopus.com/inward/record.url?scp=0001019782&partnerID=8YFLogxK

UR - http://www.scopus.com/inward/citedby.url?scp=0001019782&partnerID=8YFLogxK

U2 - 10.1016/S0040-4039(00)76177-6

DO - 10.1016/S0040-4039(00)76177-6

M3 - Article

AN - SCOPUS:0001019782

SN - 0040-4039

VL - 30

SP - 5709

EP - 5712

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 42

ER -

Mitsunobu reactions of n-alkyl and n-acyl sulfonamides-an efficient route to protected amines

Abstract

All Science Journal Classification (ASJC) codes

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