T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones

Lee J. Silverberg; Carlos Pacheco; Debashish Sahu; Peter Scholl; Hany F. Sobhi; Joshua T. Bachert; Kaitlyn Bandholz; Ryan V. Bendinsky; Heather G. Bradley; Baylee K. Colburn; David J. Coyle; Jonathon R. Dahl; Megan Felty; Ryan F. Fox; Kyanna M. Gonzalez; Jasra M. Islam; Stacy E. Koperna; Quentin J. Moyer; Duncan J. Noble; Melissa E. Ramirez; Ziwei Yang

doi:10.1002/jhet.3904

T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones

Lee J. Silverberg
, Carlos Pacheco
, Debashish Sahu
, Peter Scholl
, Hany F. Sobhi
, Joshua T. Bachert
, Kaitlyn Bandholz
, Ryan V. Bendinsky
, Heather G. Bradley
, Baylee K. Colburn
, David J. Coyle
, Jonathon R. Dahl
, Megan Felty
, Ryan F. Fox
, Kyanna M. Gonzalez
, Jasra M. Islam
, Stacy E. Koperna
, Quentin J. Moyer
, Duncan J. Noble
, Melissa E. Ramirez

Ziwei Yang

Research output: Contribution to journal › Article › peer-review

9 Scopus citations

Abstract

A series of 11 novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones was prepared at room temperature by T3P-mediated cyclization of N-aryl-C-phenyl imines with thiosalicylic acid. This provides simple and ready access to N-aryl compounds in this family, which have been generally difficult to prepare.

Original language	English (US)
Pages (from-to)	1797-1805
Number of pages	9
Journal	Journal of Heterocyclic Chemistry
Volume	57
Issue number	4
DOIs	https://doi.org/10.1002/jhet.3904
State	Published - Apr 1 2020

All Science Journal Classification (ASJC) codes

Organic Chemistry

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10.1002/jhet.3904

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Silverberg, L. J., Pacheco, C., Sahu, D., Scholl, P., Sobhi, H. F., Bachert, J. T., Bandholz, K., Bendinsky, R. V., Bradley, H. G., Colburn, B. K., Coyle, D. J., Dahl, J. R., Felty, M., Fox, R. F., Gonzalez, K. M., Islam, J. M., Koperna, S. E., Moyer, Q. J., Noble, D. J., ... Yang, Z. (2020). T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones. Journal of Heterocyclic Chemistry, 57(4), 1797-1805. https://doi.org/10.1002/jhet.3904

@article{68023336f88c46b4a4a93f5d2ff5a4df,

title = "T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones",

abstract = "A series of 11 novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones was prepared at room temperature by T3P-mediated cyclization of N-aryl-C-phenyl imines with thiosalicylic acid. This provides simple and ready access to N-aryl compounds in this family, which have been generally difficult to prepare.",

author = "Silverberg, \{Lee J.\} and Carlos Pacheco and Debashish Sahu and Peter Scholl and Sobhi, \{Hany F.\} and Bachert, \{Joshua T.\} and Kaitlyn Bandholz and Bendinsky, \{Ryan V.\} and Bradley, \{Heather G.\} and Colburn, \{Baylee K.\} and Coyle, \{David J.\} and Dahl, \{Jonathon R.\} and Megan Felty and Fox, \{Ryan F.\} and Gonzalez, \{Kyanna M.\} and Islam, \{Jasra M.\} and Koperna, \{Stacy E.\} and Moyer, \{Quentin J.\} and Noble, \{Duncan J.\} and Ramirez, \{Melissa E.\} and Ziwei Yang",

note = "Publisher Copyright: {\textcopyright} 2020 Wiley Periodicals, Inc.",

year = "2020",

month = apr,

day = "1",

doi = "10.1002/jhet.3904",

language = "English (US)",

volume = "57",

pages = "1797--1805",

journal = "Journal of Heterocyclic Chemistry",

issn = "0022-152X",

publisher = "John Wiley and Sons Inc.",

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Silverberg, LJ, Pacheco, C, Sahu, D, Scholl, P, Sobhi, HF, Bachert, JT, Bandholz, K, Bendinsky, RV, Bradley, HG, Colburn, BK, Coyle, DJ, Dahl, JR, Felty, M, Fox, RF, Gonzalez, KM, Islam, JM, Koperna, SE, Moyer, QJ, Noble, DJ, Ramirez, ME & Yang, Z 2020, 'T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones', Journal of Heterocyclic Chemistry, vol. 57, no. 4, pp. 1797-1805. https://doi.org/10.1002/jhet.3904

TY - JOUR

T1 - T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones

AU - Silverberg, Lee J.

AU - Pacheco, Carlos

AU - Sahu, Debashish

AU - Scholl, Peter

AU - Sobhi, Hany F.

AU - Bachert, Joshua T.

AU - Bandholz, Kaitlyn

AU - Bendinsky, Ryan V.

AU - Bradley, Heather G.

AU - Colburn, Baylee K.

AU - Coyle, David J.

AU - Dahl, Jonathon R.

AU - Felty, Megan

AU - Fox, Ryan F.

AU - Gonzalez, Kyanna M.

AU - Islam, Jasra M.

AU - Koperna, Stacy E.

AU - Moyer, Quentin J.

AU - Noble, Duncan J.

AU - Ramirez, Melissa E.

AU - Yang, Ziwei

PY - 2020/4/1

Y1 - 2020/4/1

N2 - A series of 11 novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones was prepared at room temperature by T3P-mediated cyclization of N-aryl-C-phenyl imines with thiosalicylic acid. This provides simple and ready access to N-aryl compounds in this family, which have been generally difficult to prepare.

AB - A series of 11 novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones was prepared at room temperature by T3P-mediated cyclization of N-aryl-C-phenyl imines with thiosalicylic acid. This provides simple and ready access to N-aryl compounds in this family, which have been generally difficult to prepare.

UR - https://www.scopus.com/pages/publications/85078786680

UR - https://www.scopus.com/pages/publications/85078786680#tab=citedBy

U2 - 10.1002/jhet.3904

DO - 10.1002/jhet.3904

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AN - SCOPUS:85078786680

SN - 0022-152X

VL - 57

SP - 1797

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JO - Journal of Heterocyclic Chemistry

JF - Journal of Heterocyclic Chemistry

IS - 4

ER -

T3P-promoted synthesis of a series of novel 3-aryl-2-phenyl-2,3-dihydro-4H-1,3-benzothiazin-4-ones

Abstract

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